| Issue Date |
Title |
Author(s) |
| 2014 |
Development of covalent inhibitors that can overcome resistance to first-generation FGFR kinase inhibitors |
Tan, Li;Wang, Jun;Tanizaki, Junko;Huang, Zhifeng;Aref, Amir R.;Rusan, Maria;Zhu, Su-Jie;Zhang, Yiyun;Ercan, Dalia;Liao, Rachel G.;Capelletti, Marzia;Zhou, Wenjun;Hur, Wooyoung;Kim, NamDoo;Sim, Taebo;Gaudet, Suzanne;Barbie, David A.;Yeh, Jing-Ruey Joanna;Yun, Cai-Hong;Hammerman, Peter S.;Mohammadi, Moosa;Jaenne, Pasi A.;Gray, Nathanael S. |
| 2015 |
Ibrutinib selectively and irreversibly targets EGFR (L858R, Del19) mutant but is moderately resistant to EGFR (T790M) mutant NSCLC Cells |
Wu, Hong;Wang, Aoli;Zhang, Wei;Wang, Beilei;Chen, Cheng;Wang, Wenchao;Hu, Chen;Ye, Zi;Zhao, Zheng;Wang, Li;Li, Xixiang;Yu, Kailin;Liu, Juan;Wu, Jiaxin;Yan, Xiao-E;Zhao, Peng;Wang, Jinhua;Wang, Chu;Weisberg, Ellen L.;Gray, Nathanael S.;Yun, Cai-Hong;Liu, Jing;Chen, Liang;Liu, Qingsong |
| 2016 |
Ibrutinib targets mutant-EGFR kinase with a distinct binding conformation |
Wang, Aoli;Yan, Xiao-E;Wu, Hong;Wang, Wenchao;Hu, Chen;Chen, Cheng;Zhao, Zheng;Zhao, Peng;Li, Xixiang;Wang, Li;Wang, Beilei;Ye, Zi;Wang, Jinhua;Wang, Chu;Zhang, Wei;Gray, Nathanael S.;Weisberg, Ellen L.;Chen, Liang;Liu, Jing;Yun, Cai-Hong;Liu, Qingsong |
| 2016 |
Pharmacological targeting of kinases MST1 and MST2 augments tissue repair and regeneration |
Fan, Fuqin;He, Zhixiang;Kong, Lu-Lu;Chen, Qinghua;Yuan, Quan;Zhang, Shihao;Ye, Jinjin;Liu, Hao;Sun, Xiufeng;Geng, Jing;Yuan, Lunzhi;Hong, Lixin;Xiao, Chen;Zhang, Weiji;Sun, Xihuan;Li, Yunzhan;Wang, Ping;Huang, Lihong;Wu, Xinrui;Ji, Zhiliang;Wu, Qiao;Xia, Ning-Shao;Gray, Nathanael S.;Chen, Lanfen;Yun, Cai-Hong;Deng, Xianming;Zhou, Dawang |
| May-2021 |
Sulfopin is a covalent inhibitor of Pin1 that blocks Myc-driven tumors in vivo |
Dubiella, Christian;Pinch, Benika J.;Koikawa, Kazuhiro;Zaidman, Daniel;Poon, Evon;Manz, Theresa D.;Nabet, Behnam;He, Shuning;Resnick, Efrat;Rogel, Adi;Langer, Ellen M.;Daniel, Colin J.;Seo, Hyuk-Soo;Chen, Ying;Adelmant, Guillaume;Sharifzadeh, Shabnam;Ficarro, Scott B.;Jamin, Yann;da Costa, Barbara Martins;Zimmerman, Mark W.;Lian, Xiaolan;Kibe, Shin;Kozono, Shingo;Doctor, Zainab M.;Browne, Christopher M.;Yang, Annan;Stoler-Barak, Liat;Shah, Richa B.;Vangos, Nicholas E.;Geffken, Ezekiel A.;Oren, Roni;Koide, Eriko;Sidi, Samuel;Shulman, Ziv;Wang, Chu;Marto, Jarrod A.;Dhe-Paganon, Sirano;Look, Thomas;Zhou, Xiao Zhen;Lu, Kun Ping;Sears, Rosalie C.;Chesler, Louis;Gray, Nathanael S.;London, Nir |
